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Antiretroviral Drugs

Fusion Inhibitors
  Enfuvirtide (Fuzeon, T-20)

Nonnucleoside Reverse Transcriptase Inhibitors (NNRTIs)
  Delavirdine (Rescriptor)
  Efavirenz (Sustiva)
  Nevirapine (Viramune)

Nucleoside Reverse Transcriptase Inhibitors (NRTIs)
  Abacavir (Ziagen)
  Abacavir + Lamivudine (Epzicom)
  Abacavir+Lamivudine+Zidovudine (Trizivir)
  Didanosine (Videx, ddI)
  Emtricitabine (Emtriva, FTC)
  Emtricitabine + Tenofovir DF (Truvada)
  Lamivudine (Epivir, 3TC)
  Lamivudine+Zidovudine (Combivir)
  Stavudine (Zerit, d4T)
  Tenofovir DF (Viread)
  Zalcitabine (Hivid, ddC)
  Zidovudine (Retrovir, AZT, ZDV)

Protease Inhibitors (PIs)
  Amprenavir (Agenerase)
  Atazanavir (Reyataz)
  Fosamprenavir (Lexiva, 908)
  Indinavir (Crixivan)
  Lopinavir+Ritonavir (Kaletra)
  Nelfinavir (Viracept)
  Ritonavir (Norvir)
  Saquinavir (Fortovase, Invirase)
Home > Drugs > Crixivan
Indinavir (Crixivan)

   Generic Name: Indinavir
    Brand Name: Crixivan

Indinavir sulfate, also known as Crixivan, is a type of antiretroviral drug called a protease inhibitor (PI). This class of drugs blocks protease, a protein that HIV needs to make more copies of itself.

AIDSinfo Drug Record for Indinavir



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Guidelines References to Indinavir

Adult and Adolescent Guidelines
Table 12a: Antiretroviral Regimens Recommended for Treatment of HIV-1 Infection in Antiretroviral Naïve Patients
Table 12b: Advantages and Disadvantages of Antiretroviral Components Recommended as Initial Antiretroviral Therapy
Table 13: Antiretroviral Dosing Recommendations for Patients with Renal or Hepatic Dysfunction
Table 14: Antiretroviral Regimens or Components That Should Not Be Offered At Any Time
Table 17: Characteristics of Protease Inhibitors (PIs)
Table 20: Drugs That Should Not Be Used With PI or NNRTI Antiretrovirals
Table 21: Drug Interactions Between Antiretrovirals and Other Drugs: PIs, NNRTIs, and NRTIs
Table 22a: Drug Effects on Blood Concentration of PIs
Table 22b: Drug Effects on Blood Concentration of NNRTIs
Table 23: HIV-Related Drugs with Overlapping Toxicities
Table 27: Suggested Minimum Target Trough Concentrations for Persons with Wild-Type HIV-1
Table 30: Preclinical and Clinical Data Concerning the Use of Antiretrovirals During Pregnancy

Pediatric Guidelines
Appendix: Characteristics of Available Antiretroviral Drugs
PI Drugs - Pediatrics
Supplement: Pediatric Antiretroviral Drug Information
Table 10: Advantages and Disadvantages of PIs for Use in Highly Active Antiretroviral Combination Regimens
Table 11: Recommended Antiretroviral Regimens for Initial Therapy for HIV Infection in Children

Perinatal Guidelines
PI Drugs - Perinatal
Table 2: Preclinical and Clinical Data Relevant to the Use of Antiretrovirals During Pregnancy
Table 3: Antiretroviral Drug Use in Pregnant HIV-Infected Women: Pharmacokinetic and Toxicity Data in Human Pregnancy and Recommendations for Use in Pregnancy

Indinavir News

Dear Healthcare Professional Letter: Changes To Labeling For Desyrel

Label Changes for Crixivan - May 2004

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More About Indinavir

AIDSinfo Drug Record for Indinavir

MEDLINEplus Fact Sheet on Indinavir

Clinical Trials Using Indinavir

Literature Citations for Indinavir

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Related Web Site Links

Join the FDA HIV/AIDS E-mail List Serv

National Library of Medicine AIDS Portal

Database for Anti-HIV Compounds

NLM - Specialized Information Services AIDSDRUGS Structures

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