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Antiretroviral Drugs

Fusion Inhibitors
  Enfuvirtide (Fuzeon, T-20)

Nonnucleoside Reverse Transcriptase Inhibitors (NNRTIs)
  Delavirdine (Rescriptor)
  Efavirenz (Sustiva)
  Nevirapine (Viramune)

Nucleoside Reverse Transcriptase Inhibitors (NRTIs)
  Abacavir (Ziagen)
  Abacavir + Lamivudine (Epzicom)
  Abacavir+Lamivudine+Zidovudine (Trizivir)
  Didanosine (Videx, ddI)
  Emtricitabine (Emtriva, FTC)
  Emtricitabine + Tenofovir DF (Truvada)
  Lamivudine (Epivir, 3TC)
  Lamivudine+Zidovudine (Combivir)
  Stavudine (Zerit, d4T)
  Tenofovir DF (Viread)
  Zalcitabine (Hivid, ddC)
  Zidovudine (Retrovir, AZT, ZDV)

Protease Inhibitors (PIs)
  Amprenavir (Agenerase)
  Atazanavir (Reyataz)
  Fosamprenavir (Lexiva, 908)
  Indinavir (Crixivan)
  Lopinavir+Ritonavir (Kaletra)
  Nelfinavir (Viracept)
  Ritonavir (Norvir)
  Saquinavir (Fortovase, Invirase)
Home > Drugs > Viracept
Nelfinavir (Viracept)

   Generic Name: Nelfinavir
    Brand Name: Viracept

Nelfinavir mesylate, also known as Viracept, belongs to the class of antiretroviral drugs called protease inhibitors (PIs). PIs act by blocking protease, a protein that HIV needs to make more copies of itself.

AIDSinfo Drug Record for Nelfinavir



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Guidelines References to Nelfinavir

Adult and Adolescent Guidelines
Table 12: Characteristics of Protease Inhibitors (PIs)
Table 14: Antiretroviral Dosing Recommendations in Patients with Renal or Hepatic Insufficiency
Table 16: Potentially Life-Threatening and Serious Adverse Events
Table 17: HIV-Related Drugs with Overlapping Toxicities
Table 18: Adverse Drug Reactions and Related "Black Box Warnings" in Product Labeling for Antiretroviral Agents
Table 19: Drugs That Should Not Be Used With PI or NNRTI Antiretrovirals
Table 20: Drug Interactions Between Antiretrovirals and Other Drugs: PIs, NNRTIs, and NRTIs
Table 21A: Drug Effects on Concentration of PIs
Table 21B: Drug Effects on Concentration of NNRTIs
Table 24: Novel Strategies To Consider For Treatment-Experienced Patients With Few Available Active Treatment Options
Table 26: Suggested Minimum Target Trough Concentrations for Persons with Wild-Type HIV-1
Table 28: Preclinical and Clinical Data Concerning the Use of Antiretrovirals During Pregnancy
Table 29: Antiretroviral Drug Use in Pregnant HIV-Infected Women: Pharmacokinetic and Toxicity Data in Human Pregnancy and Recommendations for Use in Pregnancy
Table 5: Antiretroviral Regimens Recommended for Treatment of HIV-1 Infection in Antiretroviral Naive Patients
Table 6: Advantages and Disadvantages of Antiretroviral Components Recommended as Initial Antiretroviral Therapy
Table 7: Treatment Outcome of Selected Clinical Trials of Combination Antiretroviral Regimens in Treatment-Naïve Patients with 48-Week Follow-Up Data

Pediatric Guidelines
Appendix: Characteristics of Available Antiretroviral Drugs
PI Drugs - Pediatrics
Supplement: Pediatric Antiretroviral Drug Information
Table 10: Advantages and Disadvantages of PIs for Use in Highly Active Antiretroviral Combination Regimens
Table 11: Recommended Antiretroviral Regimens for Initial Therapy for HIV Infection in Children

Perinatal Guidelines
PI Drugs - Perinatal
Table 2: Preclinical and Clinical Data Relevant to the Use of Antiretrovirals During Pregnancy
Table 3: Antiretroviral Drug Use in Pregnant HIV-Infected Women: Pharmacokinetic and Toxicity Data in Human Pregnancy and Recommendations for Use in Pregnancy

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More About Nelfinavir

AIDSinfo Drug Record for Nelfinavir

MEDLINEplus Fact Sheet on Nelfinavir

Clinical Trials Using Nelfinavir

Literature Citations for Nelfinavir

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Database for Anti-HIV Compounds

NLM - Specialized Information Services AIDSDRUGS Structures

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